| 产品名称 | Product name | CAS No. |
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洛索洛芬钠中间体 Loxoprofen Sodium Hydrate Intermediates |
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| 2-[4-(2-氧代环戊烷-1-基甲基)苯基]丙酸 | Loxoprofen | 68767-14-6 |
| 4-溴甲基苯甲酸 | 2-(4-Bromomethyl)phenylpropionic acid | 111128-12-2 |
| 2-甲氧羰基环戊酮 | Methyl 2-cyclopentanonecarboxylate | 10472-24-9 |
|
坎地沙坦酯中间体 Candesartan Cilexetil Intermediate |
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| 2-乙氧基-1-[[(2´-(1H-四唑-5-基) 联苯-4-基)甲基]苯并咪唑]-7-甲酸乙酯 | Candesartan Ethyl Ester | 139481-58-6 |
| 2-乙氧基-1-((2'-(1-三苯甲基-1H-四唑-5-基)-联苯基-4-基)甲基)-1H-苯并咪唑-7-羧酸;三苯甲基坎地沙坦 | Trityl Candesartan | 139481-72-4 |
| (±)-1-[(环己氧基)羰基氧基]乙基 2-乙氧基-1-[[2’-(1-三苯甲基-1H-四唑-5-基)联苯-4-基]甲基]-1H-苯并咪唑-7-羧酸酯;三苯甲基坎地沙坦酯 | Trityl Candesartan Cilexetil | 170791-09-0 |
|
格列吡嗪中间体 Glipizide Intermediates |
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| 4-[2-(5-甲基吡嗪-2-甲酰氨基)乙基]苯磺酰胺 | 4-[β-(5-Methylpyrazinyl-2-carboxamido)ethyl]benzene Sulfonamide | 33288-71-0 |
| [[4–[2-(5-甲基吡嗪-2-酰胺基)乙基]苯基]磺酰基]氨基甲酸乙酯 | ethyl N-[4-[2-[(5-methylpyrazine-2-carbonyl)amino]ethyl]phenyl]sulfonylcarbamate | 1076198-09-8 |
| (乙氧羰基)(4-(2-(5-甲基吡嗪-2-甲酰胺)乙基)苯基)磺酰胺环己基铵盐 | (ethoxycarbonyl)(4-(2-(5-methylpyrazine-2-formamide) ethyl) phenyl) sulfonamide cyclohexyl ammonium salt | — |
| 5-甲基吡嗪-2-羧酸 | 5-Methylpyrazine-2-carboxylic acid | 5521-55-1 |
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盐酸特拉唑嗪中间体 Terazosin Intermediate |
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| N-(2-四氢呋喃甲酰基)哌嗪 | 1-(Tetrahydro-2-furoyl)piperazine | 63074-07-7 |
| 1-(4-氨基-6,7-二甲氧基-2-喹唑啉基)-4-[(四氢呋喃-2-甲酰基)哌嗪 | [4-(4-amino-6,7-dimethoxyquinazolin-2-yl)piperazin-1-yl]-(oxolan-2-yl)methanone | 63590-64-7 |
| 2-氯-4-氨基一6,7-二甲氧基喹唑啉 | 4-Amino-2-chloro-6,7-dimethoxyquinazoline | 23680-84-4 |
| 2-四氢糠酸 | 2-Tetrahydrofuroic acid | 16874-33-2 |
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硝苯地平中间体 Nifidipine Intermediate |
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| 3-氨基巴豆酸甲酯 | Methyl 3-aminocrotonate | 14205-39-1 |
| 2-(2-硝基苯亚甲基)乙酰乙酸甲酯 | Methyl 3-nitrobenzylideneacetoacetate | 39562-17-9 |
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奥美沙坦酯中间体 Olmesartan Intermediate |
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| 4-(1-羟基-1-甲基乙基)-2-丙基-1-[[2’-[2-(三苯基甲基)-2H-四氮唑-5-基]联苯-4-基]甲基]咪唑-5-羧酸乙酯 | Ethyl 4-(2-hydroxy-2-propanyl)-2-propyl-1-{[2'-(1-trityl-1H-tetra zol-5-yl)-4-biphenylyl]methyl}-1H-imidazole-5-carboxylate | 144690-33-5 |
| 4-(1-羟基-1-甲基乙基)-2-丙基-1-[[2’-[2-(三苯基甲基)-2H-四氮唑-5-基]联苯-4-基]甲基]咪唑-5-羧酸 | Trityl Olmesartan Acid | 761404-85-7 |
| (5-甲基-2-氧代-1,3-二氧环戊烯-4-基)甲基 4-(1-羟基-1-甲基乙基)-2-丙基-1-[[2’-[2-(三苯基甲基)-2H-四氮唑-5-基]联苯-4-基]甲基]咪唑-5-甲酸酯 | (5-methyl-2-oxo-1,3-dioxol-4-yl)methyl 5-(2-hydroxypropan-2-yl)-2-propyl-3-[[4-[2-(2-trityltetrazol-5-yl)phenyl]phenyl]methyl]imidazole-4-carboxylate | 1020157-01-0 |
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塞来昔布中间体 celecoxib Intermediate |
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| 4-磺酰胺基苯肼盐酸盐 | 4-Sulfonamide-phenylhydrazine hydrochloride | 27918-19-0 |
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替米沙坦中间体 Telmisartan Intermediates |
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| 2-正丙基-4-甲基-6-(1′-甲基苯并咪唑-2-基)苯并咪唑 | 2-n-propyl-4-methyl-6-(1-methylbenzimidazole-2-ly)benzimidazole | 152628-02-9 |
| 4'-溴甲基联苯-2-甲酸甲酯 | Methyl4'-bromomethyl biphenyl-2-carboxylate | 114772-38-2 |
| 4'-甲基联苯-2-甲酸甲酯 | Methyl 4'-methylbiphenyl-2-carboxylate | 114772-34-8 |
| 2-正丙基-4-甲基-6-羧基苯并咪唑 | 4-methyl-2-propyl-1H-Benzimidazole-6-carboxylic acid | 152628-03-0 |
|
双咪唑起始物料 2-n-propyl-4-methyl-6-(1-methylbenzimidazole-2-ly)benzimidazole Starting material |
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| 3-甲基-4-氨基苯甲酸 | 4-Amino-3-methylbenzoic acid | 2486-70-6 |
| 3-甲基-4-硝基苯甲酸 | 3-Methyl-4-nitrobenzoic acid | 3113-71-1 |
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非布司他中间体 Febuxostat Intermediate |
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| 2-(3-醛基-4-异丁氧基苯基)-4-甲基噻唑-5-甲酸乙酯 | Ethyl 2-(3-formyl-4-isobutoxyphenyl)-4-methylthiazole-5-carboxylate | 161798-03-4 |
| 2-(3-氰基-4-异丁氧基苯基)-4-甲基噻唑-5-甲酸乙酯 | Ethyl 2-(3-cyano-4-isobutoxyphenyl)-4-methylthiazole-5-carboxylate | 160844-75-7 |
| 2-[(3-氰基-4-异丁氧基)苯基]-4-甲基-5-噻唑羧酸 | 2-[(3-cyano-4-isobutoxy)phenyl] -4-methyl-5-thiazolcarboxylic acid | 144060-53-5 |
| 2-(3-醛基-4-羟基苯基)-4-甲基噻唑-5-羧酸乙酯 | Ethyl 2-(3-formyl-4-hydroxyphenyl)-4-methylthiazole-5-carboxylate | 161798-01-2 |
|
他达拉非中间体 Tadalafil Intermediate |
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| ((1R,3R)-1-(1,3-苯并二氧戊环-5-基)-2-(氯乙酰基)-2,3,4,9-四氢-1H-吡啶并[3,4-B]吲哚-3-羧酸甲酯) | Methyl (1R,3R)-1-(1,3-benzodioxol-5-yl)-2-(chloroacetyl)-2,3,4,9-tetrahydro-1H-β-carboline-3-carboxylate | 171489-59-1 |
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盐酸多奈哌齐中间体 Donepezil Intermediate |
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| ( 5,6-二甲氧基-2-(4-吡啶基)亚甲基-1-茚酮) | 5,6-Dimethoxy-2-(pyridine-4-yl)methylene-indan-1-one | 4803-74-1 |
|
枸橼酸西地那非中间体 Sildenafil Citrate Intermediate |
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| 2-乙氧基-5-((4-甲基哌嗪-1-基)磺酰基)苯甲酸 | 2-ethoxy-5-(4-methylpiperazin-1-yl)sulfonylbenzoic acid | 194602-23-8 |
| 4-氨基-1-甲基-3-丙基-1H-吡唑-5-甲酰胺盐酸盐 | 4-Amino-1-methyl-3-propyl-1H-pyrazole-5-carboxamide Hydrochloride | 247584-10-7 |
| 4-(2-乙氧基-5-((4-甲基哌嗪-1-基)磺酰基)苯甲酰胺基)-1-甲基-3-丙基-1H-吡唑-5-甲酰胺 | 4-{2-ethoxy-5-[(4-methylpiperazin-1-yl)sulfonyl]benzamido}-1-methyl-3-propyl-1H-pyrazole-5-carboxamide | 200575-15-1 |
| 1-{4-乙氧基-3-(6,7-二氢-1-甲基-7-氧代-3-丙基-1氢-吡唑并[4,3d]喀啶-5-基)苯磺酰}-4-甲基哌嗪 | 5-{2-ethoxy-5-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}-1-methyl-3-propyl-1H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one | 139755-83-2 |
| 4-(2-乙氧基苯甲酰胺)-1-甲基-3-正丙基吡唑-5-甲酰胺 | 4-(2-ethoxy benzamido)-1-methyl-3-n-propyl pyrazole-5-carboxamide. | 139756-03-9 |
| 5-(2-乙氧苯基)-1-甲基-3-丙基-1,6-二氢-7H-吡唑并[4,3-D]嘧啶-7-酮 | 5-(2-ethoxyphenyl)-1-methyl-3-n-propyl-1,6-dihydro-7h-pyrazolo[4,3-d]-7-pyrimidinon | 139756-21-1 |
|
右佐匹克隆中间体 Dexzopiclone intermediate |
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| (5RS)-6-(5-氯吡啶-2-基)-7-[(4-甲基哌嗪-1-基)羰氧基]-5,6-二氢吡咯并[3,4-b]吡嗪-5-酮 | zopiclone | 43200-80-2 |
| (+)-(7S)-6-(5-氯-2-吡啶基)-7-[(4-甲基哌嗪-1-基)甲酰氧基]-5,6-二氢吡咯并[3,4-b]吡嗪-5-酮-D-二苯甲酰酒石酸盐 | D(+)-O,O-dibenzoyl tartarate of zopiclone | 1020156-02-8 |
| 4-甲基哌嗪-1-甲酰氯盐酸盐 | 4-Methyl-1-piperazinecarbonyl chloride hydrochloride | 55112-42-0 |
| 6-(5-氯-2-吡啶基)-6,7-二氢-7-羟基-5H-吡咯并[3,4-b]吡嗪-5-酮 | 6-(5-Chloro-2-pyridyl)-6,7-dihydro-7-hydroxy-5H-pyrrolo[3,4-b]pyrazin-5-one | 43200-81-3 |
|
利伐沙班中间体 Rivaroxaban Intermediate |
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| (2-[(2R)-2-羟基-3-[[4-(3-氧代-4-吗啉基)苯基]氨基]丙基]-1H-异吲哚-1,3(2H)-二酮) | 4-[((2R)-Hydroxy-3-phthalimido)propylamine]phenyl-3-morpholinone | 446292-07-5 |
| (2-[[(5S)-2-氧代-3-[4-(3-氧代-4-吗啉基)苯基]-5-噁唑烷基]甲基]-1H-异吲哚-1,3(2H)-二酮) | 2-[[(5S)-2-Oxo-3-[4-(3-oxo-4-morpholinyl)phenyl]-5-oxazolidinyl]methyl]-1H-isoindole-1,3(2H)-dione | 446292-08-6 |
| (4-[4-[(5S)-5-(氨基甲基)-2-氧代-3-恶唑烷基]苯基]-3-吗啉酮盐酸盐) | (S)-4-(4-(5-(Aminomethyl)-2-oxooxazolidin-3-yl)phenyl)morpholin-3-one hydrochloride | 898543-06-1 |
|
阿哌沙班中间体 apixaban Intermediate |
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| 5-氯-N-(4-(3-吗啉-2-氧代-5,6-二氢吡啶-1(2H)-基)苯基)戊酰胺 | 5-Chloro-N-[4-[5,6-dihydro-3-(4-morpholinyl)-2-oxo-1(2H)-pyridinyl]phenyl]pentanamide | 1643330-62-4 |
| 5,6-二氢-3-(4-吗啉基)-1-[4-(2-氧代-1-哌啶基)苯基]-2(1H)-吡啶酮 | 5,6-Dihydro-3-(4-morpholinyl)-1-[4-(2-oxo-1-piperidinyl)phenyl]-2(1H)-pyridinone | 545445-44-1 |
| 1-(4-甲氧基苯基)-7-氧代-6-(4-(2-氧代哌啶-1-基)苯基)-4,5,6,7-四氢-1H-吡唑[3,4-c]吡啶-3-甲酸乙酯 | 1-(4-methoxy-phenyl)-7-oxo-6-[4-(2-oxo-piperidin-1-yl)-phenyl]-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxylic acid ethyl ester | 503614-91-3 |
|
格列喹酮中间体 Gliquidone Intermediate |
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| 7-甲氧基-2,4,4-三甲基-异喹啉-1,3(2H,4H)-二酮 | 7-Methoxy-2,4,4-trimethylisoquinoline-1,3-(2H,4H)-dione | 191988-38-2 |
| 7-甲氧基-4,4-二甲基-异苯并吡喃-1,3-二酮 | 7-methoxy-4,4-dimethylisochromene-1,3-dione | 55974-25-9 |
| 4-[2-(7-甲氧基-4,4-二甲基-1,3-二酮-3,4- 二氢异喹啉-2(1H)-基)乙基]苯磺酰胺 | 4-(2-(3,4-dihydro-7-methoxy-4,4-dimethyl- 1,3-dioxo-2(1h)-isoquinolinyl)ethyl) benzenesulfonamide | 33456-68-7 |
| 3-三氯甲基-6-甲氧基-1(3H)-异构苯并呋喃酮 | 3-trichloromethyl-6-methoxy-1 (3H) -isobenzofuranone | — |
| 2-(β,β-二氯乙烯基)-5-甲氧基苯甲酸 | 2- (β, β-dichloroethylene) -5-methoxybenzoic acid | — |
| 2-羧甲基-5-甲氧基苯甲酸 | 2-(carboxymethyl)-5-methoxybenzoic acid | 52962-25-1 |
| 7-甲氧基-2-甲基-异喹啉-1,3(2H,4H)-二酮 | 4-methoxy-N-methylhomophthalimide | 76746-95-7 |
|
沙库比曲缬沙坦钠中间体 Valsartan-Sacubitril Intermediate |
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| (R,E)-乙基 5-([1,1'-联苯]-4-基)-4-((叔丁氧羰基)氨基)-2-甲基-2-戊烯酸 | ethyl 5-(4-[1,1'-biphenyl]yl)-4-[[(1,1-dimethylethoxy)carbonyl]amino]-2-methyl-2-pentenoate | 149709-59-1 |
| (R,E)-5-([1,1'-联苯]-4-基)-4-((叔丁氧羰基)氨基)-2-甲基-2-戊烯酸 | (R,E)-5-([1,1'-biphenyl]-4-yl)-4-((tert-butoxycarbonyl)amino)-2-methylpent-2-enoic acid | 1012341-48-8 |
| ((2R,4S)-5-([1,1'-联苯]-4-基)-4-((叔丁氧羰基)氨基)-2-甲基戊酸) | (2R,4S)-5-(Biphenyl-4-yl)-4-[(tert-butoxycarbonyl)amino]-2-methylpentanoic acid | 1012341-50-2 |
| ((2R,4S)-乙基 5-([1,1'-联苯]-4-基)-4-氨基-2-甲基戊酸盐酸盐) | (2R,4S)-ethyl 5-([1,1'-biphenyl]-4-yl)-4-amino-2-methylpentanoate hydrochloride | 149690-12-0 |
| ((2R,4S)-5-(联苯-4-基)-4-(氨基)-5-(3-羧基-丙酰基氨基)-2-甲基-戊酸乙酯钙盐) | Ethyl (2R,4S)-5-(Biphenyl-4-yl)-4-(amino)-5-(3-carboxypropionyl)amino]-2-methylpentanoate, calcium salt | 1369773-39-6 |
|
沙库比曲缬沙坦钠中间体(D-N-BOC联苯丙氨醇)起始物料 Valsartan-Sacubitril Intermediate Starting material |
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| 3-联苯基-4-基-2-氧代丙酸 | 3-(4-Biphenylyl)pyruvic acid | 91853-46-2 |
| (R)-2-氨基-3-联苯基-4-基丙酸 (D-联苯丙氨酸) | D-4,4'-Biphenylalanine | 170080-13-4 |
| (R)-2-氨基-3-联苯基-4-基-丙酸甲酯盐酸盐 | methyl (2R)-2-amino-3-(4-phenylphenyl)propanoate | 169885-19-2 |
| (R)-3-联苯-4-基-2-叔丁氧羰基氨基丙酸甲酯 | methyl (2R)-2-[(2-methylpropan-2-yl)oxycarbonylamino]-3-(4-phenylphenyl)propanoate | 149818-98-4 |
| (R)-叔丁基(1-([1,1’-联苯]-4-基)-3-羟基丙烷-2-氨基甲酸酯 | N-[(1R)-2-[1,1'-Biphenyl]-4-yl-1-(hydroxymethyl)ethyl]carbamic acid 1,1-dimethylethyl ester | 1426129-50-1 |
|
阿齐沙坦中间体 Azilsartan Intermediate |
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| 2-[[(2'-氰基联苯-4-基)甲基]氨基]-3-硝基苯甲酸乙酯 | Ethyl-2-[[(2'-cyanobiphenyl-4-yl)methyl]amino]-3-nitrobenzoate | 136285-67-1 |
| 3-氨基-2-[(2'-氰基联苯-4-基)甲基]氨基苯甲酸乙酯 | ethyl 3-amino-2-[[4-(2-cyanophenyl)phenyl]methylamino]benzoate | 136285-69-3 |
| 2-乙氧基-1-[[(2'-腈基连苯-4-取代)甲基]苯并咪唑]-7-羧酸乙酯 | Ethyl-2-Ethoxy-1-[[(2'-Cyanobiphenyl-4-yl) Methyl] Benzimidazole]-7-Carboxylate | 139481-41-7 |
| 2-乙氧基-1-[[2'-(羟基脒基)联苯基-4-基]甲基]-1H-苯并咪唑-7-甲酸甲酯 | 2-Ethoxy-1-[[2'-[(hydroxyamino)iminomethyl][1,1'-biphenyl]-4-yl]methyl]-1H-benzimidazole-7-carboxylic acid methyl ester | 147403-65-4 |
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孟鲁司特钠中间体 Montelukast sodium intermediate |
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| (R-(E))-1-(((1-(3-(2-(7-氯-2-喹啉基)乙烯基)苯基)-3-(2-(1-羟基-1-甲基乙基)苯基)丙基)硫)甲基)环丙基乙酸; | Montelukastl | 158966-92-8 |
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琥珀酸索利那新中间体 Solifenacin succinate Intermediate |
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| (S)-1-苯基-3,4-二氢异喹啉-2-(1H)-甲酰氯 | (S)-1-phenyl-3,4-dihydro-1H-isoquinoline-2-carbonyl chloride | 1195949-26-8 |
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盐酸托莫西汀中间体 Atomoxetine Intermediate |
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| 3-甲氨基-1-苯基-1-丙酮盐酸盐 | 3-(methylamino)-1-phenylpropan-1-one,hydrochloride | 2538-50-3 |
| 3-N-甲基-1-苯基丙醇 | 3-Hydroxy-N-Methyl-3-Phenyl-Propylamine | 42142-52-9 |
| N-甲基-3-(2-甲基苯氧基)-3-苯基丙胺草酸盐 | N,N-Dimethyl-3-(o-tolyloxy)-3-phenylpropylamine | 83015-25-2 |
| N-甲基-3-(2-甲基苯氧基)-3-苯基丙胺-L-酒石酸盐 | N-methyl-3 - (2-methylphenoxy) -3-phenylpropylamine - L-tartrate | — |
|
利格列汀中间体 Linagliptin Intermediate |
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| (R)-2-(3-哌啶基)异吲哚-1,3-二酮盐酸盐 | (R)-2-(piperidin-3-yl)isoindoline-1,3-dione hydrochloride | 1381795-31-8 |
| 8-溴-7-(2-丁炔基)-3,7-二氢-3-甲基-1H-嘌呤-2,6-二酮 | 8-Bromo-7-(but-2-yn-1-yl)-3-methyl-1H-purine-2,6(3H,7H)-dione | 666816-98-4 |
| 8-溴-7-(2-丁炔基)-3-甲基-1-((4-甲基-2-喹唑啉基)甲基)-3,7-二氢-1H-嘌呤-2,6-二酮 | 8-bromo-7-but-2-ynyl-3-methyl-1-[(4-methylquinazolin-2-yl)methyl]purine-2,6-dione | 853029-57-9 |
| (R)-7-2-丁炔基)-8-(3-(1,3-二氧异吲哚)哌啶基)-3-甲基-1-((4-甲基-2-喹唑啉基)甲基)-3,7-二氢-1H-嘌呤-2,6-二酮 | 1H-Purine-2,6-dione, 7-(2-butyn-1-yl)-8-[(3R)-3-(1,3-dihydro-1,3-dioxo-2H-isoindol-2-yl)-1-piperidinyl]-3,7-dihydro-3-methyl-1-[(4-methyl-2-quinazolinyl)methyl]- | 886588-63-2 |
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富马酸伏诺拉生中间体 Vonoprazan Fumarate Intermediate |
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| 2-[2-(2-氟苯基)-2-氧代乙基]丙二腈 | 2-[2-(2-Fluorophenyl)-2-oxoethyl]propanedinitrile | 312307-38-3 |
| 5-(2-氟苯基)-1H-吡咯-3-腈 | 5-(2-fluorophenyl)-1H-pyrrole-3-carbonitrile | 1240948-77-9 |
| 5-(2-氟苯基)-1H-吡咯-3-甲醛 | 5-(2-fluorophenyl)-1H-pyrrole-3-carbaldehyde | 881674-56-2 |
| 5-(2-氟苯基)-1-(吡啶-3-磺酰基)-1H-吡咯-3-甲醛 | 5-(2-fluorophenyl)-1-(pyridine-3-sulfonyl)-1H-pyrrole-3-carbaldehyde | 881677-11-8 |
| 1-(5-(2-氟苯基)-1-(吡啶-3-基磺酰)-1H-吡咯-3-基)-N-甲基甲胺富马酸盐 | 1-(5-(2-fluorophenyl)-1-(pyridine-3-yl sulfonyl) -1H-pyrrole-3-yl) -N-methylmethylamine fumarate | 2098974-13-9 |
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盐酸伊托必利中间体 Itopride Hydrochloride Intermediate |
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| (4-(2-(二甲胺基)乙氧基)苯腈 | 4-[2-(dimethylamino)ethoxy]benzonitrile | 24197-95-3 |
| (4-(2-(二甲胺基)乙氧基)苄胺 | 2-[4-(aminomethyl)phenoxy]-N,N-dimethylethanamine | 20059-73-8 |
| N-(4-(2-(二甲胺基)乙氧基)苯甲基)-3,4-二甲氧基苯甲酰胺 | N-[[4-[2-(dimethylamino)ethoxy]phenyl]methyl]-3,4-dimethoxybenzamide | 122898-67-3 |
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盐酸鲁拉西酮中间体 Lurasidone Hydrochloride Intermediate |
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| (3aR,7 aR)-4’-(苯并[ d ]异噻唑 -3-基)八氢螺旋[异吲哚 -2,1’ -哌嗪] -2-甲基磺酸铵 | 4-(1,2-Benzothiazol-3-yl)-1-[(3aR,7aR)-octahydro-2H-isoindol-2-yl ]piperazin-1-ium-1-sulfonate | 186204-37-5 |
| (3aR,4 S,7 R,7 aS)-2-((1R,2 R)-2-(4-(苯并 [ d ]异噻唑 -3-基)哌嗪 -1-甲基)环己基)甲基)六氢 -1H-4,7-甲基异吲哚 -1,3(2H)-二酮 | lurasidone | 367514-87-2 |
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格列美脲中间体 Glimepiride Intermediate |
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| 3-乙基-4-甲基-3-吡咯啉-2-酮-1-羧酸苯酯 | 3-ethyl-4-methyl-3-pyrrolin-2-keto-1-carboxylate phenyl ester | 2128304-88-9 |
| 4-[2-(3-乙基-4-甲基-2-氧代-3-吡咯啉-1-甲酰氨基)乙基]苯磺酰胺 | 4-[2-[(3-Ethyl-4-methyl-2-oxo-3-pyrrolin-1-yl)carboxamido]ethyl]benzenesulfonamide | 119018-29-0 |
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琥珀酸曲格列汀中间体 Trelagliptin Succinate Intermediate |
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| 2-氰基-5-氟溴苄 | 2-Cyano-5-Fluorobenzyl Bromide | 421552-12-7 |
| 2-[(6-氯-3,4-二氢-3-甲基-2,4-二氧代-1(2H)-嘧啶基)甲基] -4-氟苯甲腈 | 2-[(6-chloro-3,4-dihydro-3-methyl-2,4-dioxo-1(2H)-pyrimidinyl)methyl]-4-fluorobenzonitrile | 865759-24-6 |
| 2-[[6-[(3R)-3-氨基-1-哌啶基]-3,4-二氢-3-甲基-2,4-二氧代-1(2H)-嘧啶基]甲基]-4-氟苯甲腈 | Trelagliptin | 865759-25-7 |
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米拉贝隆中间体 Mirabegron intermediates |
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| 2-氨基-4-噻唑乙酸乙酯 | Ethyl 2-amino-4-thiazoleacetate | 53266-94-7 |
| 2-氨基噻唑-4-乙酸 | 2-(2-amino-1,3-thiazol-4-yl)acetic acid | 29676-71-9 |
| (R)-N-(4-硝基苯乙基)-2-羟基-2-苯基乙酰胺 | (2R)-2-Hydroxy-N-[2-(4-nitrophenyl)ethyl]-2-phenylacetamide | 521284-19-5 |
| (R)-2-(4-硝基苯乙基氨基)-1-苯基乙醇盐酸盐 | (1R)-2-[2-(4-nitrophenyl)ethylamino]-1-phenylethanol,hydrochloride | 521284-21-9 |
| (R)-[[[2-(4-氨基苯基)乙基]氨基]甲基]-苯甲醇盐酸盐 | (R)- [[[2- (4-aminophenyl) ethyl] amino] methyl] - benzyl alcohol hydrochloride | 521284-22-0 |
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恩格列净中间体 Empagliflozin intermediates |
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| (3R,4S,5R,6R)-3,4,5-三(三甲基硅氧基)-6-((三甲基硅氧基)甲基)四氢-2H-吡喃-2-酮 | (3R,4S,5R,6R)-3,4,5-tris(trimethylsilyloxy)-6-(trimethylsilyloxymethyl)oxan-2-one | 32384-65-9 |
| 三乙酸(2R,3R,4R,5S,6S)-2-(乙酰氧基甲基)-6-(4-氯-3-(4-((S)-四氢呋喃-3-基氧基)苄基)苯基)四氢-2H-吡喃-3,4,5 | (1S)-1,5-anhydro-2,3,4,6-tetra-O-acteyl-1-C-[4-chloro-3-[[4-[[(3S)-tetrahydrofu-ran-3-yl]oxy]phenyl] methyl]phenyl]-D-Glucitol | 915095-99-7 |
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美阿沙坦钾中间体 Azilsartan Medoxomil intermediate |
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| 4-甲酰氧基-5-甲基-1,3-二氧杂环戊烯-2-酮 | 4-formyloxy-5-methyl-1, 3-dioxole-2-one | 209551-67-7 |
| 4-羟甲基-5-甲基-1,3-二氧杂环戊烯-2-酮 | 4-(Hydroxymethyl)-5-methyl-1,3-dioxol-2-one | 91526-18-0 |
| 1-[(2'-(N'-羟基甲脒基)[1,1'-联苯基]-4-基)甲基]-2-乙氧基-1H-苯[d]咪唑-7-羧酸乙酯 | ethyl 2-ethoxy-1-((2′-(N′-hydroxycarbamimidoyl)biphenyl-4-yl)methyl)-1H-benzo[d]imidazole-7-carboxylate | 1397836-41-7 |
| 2-乙氧基-1-[[2'-(5-氧代-4,5二氢-1,2,4-噁二唑-3-基)联苯-4-基]甲基]-1H-苯并咪唑-7-羧酸 | azilsartan | 147403-03-0 |
| 2-乙氧基-1-[2'-(5-氧代-l, 2, 4-噁二唑-3-基)联苯-4-甲基]苯并咪唑-7-[(5-甲基-2-氧代-1,3-间二氧杂环戊烯-4-基)甲基]羧酸酯 | azilsartan medoxomil | 863031-21-4 |
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依折麦布中间体 Ezetimibe intermediate |
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| 4-[[(4-氟苯基)亚胺]甲基]-苯酚 | 4-[[(4-Fluorophenyl)imino]methyl]-phenol | 3382-63-6 |
| (4S)-3-[(2R,5S)-5-(4-氟苯基)-2-[(S)-[(4-氟苯基)氨基]({4-[(三甲基硅)氧]苯基})甲基]-5-[(三甲基硅)氧]正戊酰基]-4-苯基-1,3-恶唑烷-2-酮 | (4S)-3-[(2R,5S)-5-(4-fluorophenyl)-2-[(S)-[(4-fluorophenyl)amino]-(4-trimethylsilyloxyphen yl)methyl]-5-trimethylsilyloxy-pentanoyl]-4-phenyl-1,3-oxazolidin-2-one | 272778-12-8 |
| (4S)-3-[5-(4-氟苯基)-1,5-二氧代戊基]-4-苯基-2-恶唑烷酮 | 1-(4-fluorophenyl)-5-[(4S)-2-oxo-4-phenyl-1,3-oxazolidin-3-yl]pentane-1,5-dione | 189028-93-1 |
| 4-(4-氟苯甲酰基)丁酸 | 4-(4-Fluorobenzoyl)Butyric Acid | 149437-76-3 |
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磷酸奥司他韦中间体 Oseltamivir Phosphate intermediate |
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| (3R,4S,5R)-5-(叔丁基氨基)-4-羟基-3-(戊烷-3-基氧基)环己-1-烯-1-羧酸乙酯 | ethyl (3R,4S,5R)-5-N-(1,1-dimethylethyl)amino-3-(1-ethylpropoxy)-4-hydroxy-1-cyclohexene-1-carboxylate | 651324-04-8 |
| (1R,5R,6R)-7-叔丁基-5-(戊烷-3-氧基)-7-氮杂双环[4.1.0]庚-3-烯-3-羧酸乙酯 | (1 r, 5 r, 6 r) - 7 - tert-butyl - 5 - (pentane - 3 - oxygen radicals) - 7 - nitrogen mixed double loop - 3 - [4.1.0] g ene - 3 - carboxylic acid ethyl ester | 2417645-75-9 |
| (3R,4R,5S)-4-(叔丁基氨基)-5-(二烯丙胺基)-3-(戊烷-3基氧基)环己-1-烯-1-羧酸乙酯二盐酸盐 | (3 r, 4 r, 5 s) - 4 - (butylated amino) - 5 - (diallyl amino) - 3 - (pentane - 3 oxo) cyclohexanol - 1 - ene - 1 - carboxylic acid ethyl ester hydrochloride | — |
| (3R,4R,5S)-4-N-乙酰基(叔丁基)氨基-5-N,N-二烯丙基氨基-3-(1-乙基丙氧基)-1-环己烯-1-甲酸乙酯单盐酸盐 | ethyl (3R,4R,5S)-4-[acetyl(tert-butyl)amino]-5-[bis(prop-2-enyl)amino]-3-pentan-3-yloxycyclohexene-1-carboxylate,hydrochloride | 651324-08-2 |
| (3R,4R,5S)-4-乙酰氨基-5-(二烯丙基氨基)-3-(戊-3-基氧基)环己-1-烯甲酸乙酯 | Ethyl (3R,4R,5S)-4-N-Acetylamino-5-N,N-diallylamino-3-(1-ethylpropoxy)-1-cyclohexene-1-carboxylate | 651324-09-3 |
| (3R,4R,5S)-4-乙酰胺基-5-氨基-3-(1-乙基丙氧基)-1-环己烯-1-甲酸乙酯 | oseltamivir | 196618-13-0 |
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拉考沙胺中间体 lacosamide intermediate |
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| (2R)-2-叔丁氧羰基氨基-N-苄基-3-羟基丙酰胺 | Boc-Ser-NHCH2C6H5 | 141108-78-3 |
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普瑞巴林中间体 Pregabalin intermediate |
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| 3-异丁基戊二酰亚胺 | 3-Isobutylpiperidine-2,6-dione | 916982-10-0 |
| (R)-3-(氨甲酰甲基)-5-甲基己酸 | R-(-)-3-(Carbamoylmethyl)-5-methylhexanoic acid | 181289-33-8 |
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匹伐他汀钙中间体 Pivastatin calcium intermediate |
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| (4R,6S)-6-[[(1E)-2-环丙基-4-(4-氟苯基)-3-喹啉基]乙烯基]-2,2-二甲基-1,3-二氧六环-4-乙酸叔丁酯 | (4R,6S)-6-[(1E)-2-[2-Cyclopropyl-4-(4-fluorophenyl)-3-quinolinyl]ethenyl]-2,2-dimethyl-1,3-dioxane-4-acetic acid tert-butyl ester | 147489-06-3 |
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硫酸氨基葡萄糖氯化钠复盐 Glucosamine sulfate intermediate |
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| 硫酸氨基葡萄糖氯化钠复盐 | Glucosamine sulfate sodium chloride double salt | 1296149-13-7 |
| 瑞舒伐他汀钙中间体 | ||
| 2-[(4R,6S)-6-[(E)-2-[4-(4-氟苯基)-6-异丙基-2-(N-甲基-N-甲磺酰氨基)嘧啶-5-基]乙烯基]-2,2-二甲基-1,3-二氧六环-4-基]乙酸叔丁酯 | tert-Butyl 6-[(1E)-2-[4-(4-fluorophenyl)-6-(1-methylethyl)-2-[methyl(methylsulfonyl)amino]-5-pyrimidinyl]ethenyl]-2,2-dimethyl-1,3-dioxane-4-acetate | 289042-12-2 |
| (E)-7-[4-(4-氟基苯基)-6-异丙基-2-[甲基(甲磺酰基)氨基]-嘧啶-5-基]-(3R,5S)-3,5-二羟基庚-6-烯酸叔丁酯 | (3R,5S,6E)-7-[4-(4-Fluorophenyl)-6-isopropyl-2-[(methanesulfonyl) methylamino]pyrimidin-5-yl]-3,5-dihydroxyhept-6-enoic acid tert-butyl ester | 355806-00-7 |
